| Design of novel and selective inhibitors of urokinase-type plasminogen activator with improved pharmacokinetic properties for use as antimetastatic agents A Schweinitz, T Steinmetzer, IJ Banke, MJE Arlt, A Sturzebecher, ... Journal of Biological Chemistry 279 (32), 33613-33622, 2004 | 167 | 2004 |
| Crystals of the urokinase type plasminogen activator variant βc-uPA in complex with small molecule inhibitors open the way towards structure-based drug design E Zeslawska, A Schweinitz, A Karcher, P Sondermann, S Sperl, ... Journal of molecular biology 301 (2), 465-475, 2000 | 91 | 2000 |
| Crystals of urokinase type plasminogen activator complexes reveal the binding mode of peptidomimetic inhibitors E Zeslawska, U Jacob, A Schweinitz, G Coombs, W Bode, E Madison Journal of molecular biology 328 (1), 109-118, 2003 | 48 | 2003 |
| The 5-aromatic hydantoin-3-acetate derivatives as inhibitors of the tumour multidrug resistance efflux pump P-glycoprotein (ABCB1): Synthesis, crystallographic and biological … E Żesławska, A Kincses, G Spengler, W Nitek, K Wyrzuc, ... Bioorganic & Medicinal Chemistry 24 (12), 2815-2822, 2016 | 35 | 2016 |
| Highly efficient microwave synthesis of rhodanine and 2-thiohydantoin derivatives and determination of relationships between their chemical structures and antibacterial activity W Tejchman, B Orwat, I Korona-Głowniak, A Barbasz, I Kownacki, ... RSC advances 9 (67), 39367-39380, 2019 | 28 | 2019 |
| Pronounced activity of aromatic selenocyanates against multidrug resistant ESKAPE bacteria MJ Nasim, K Witek, A Kincses, AY Abdin, E Żesławska, MA Marć, ... New Journal of Chemistry 43 (15), 6021-6031, 2019 | 27 | 2019 |
| Structural analysis and antimicrobial activity of 2 [1H]-pyrimidinethione/selenone derivatives E Żesławska, I Korona-Głowniak, M Szczesio, A Olczak, A Żylewska, ... Journal of Molecular Structure 1142, 261-266, 2017 | 25 | 2017 |
| Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH3 or 2-CH3 A Gunia-Krzyżak, D Żelaszczyk, A Rapacz, E Żesławska, ... Bioorganic & Medicinal Chemistry 25 (2), 471-482, 2017 | 21 | 2017 |
| N-[(2, 6-Dimethylphenoxy) alkyl] aminoalkanols—their physicochemical and anticonvulsant properties AM Waszkielewicz, M Cegła, E Żesławska, W Nitek, K Słoczyńska, ... Bioorganic & Medicinal Chemistry 23 (15), 4197-4217, 2015 | 20 | 2015 |
| Computer-aided insights into receptor-ligand interaction for novel 5-arylhydantoin derivatives as serotonin 5-HT7 receptor agents with antidepressant activity K Kucwaj-Brysz, R Kurczab, M Jastrzębska-Więsek, E Żesławska, ... European Journal of Medicinal Chemistry 147, 102-114, 2018 | 18 | 2018 |
| Anticonvulsant activity, crystal structures, and preliminary safety evaluation of N-trans-cinnamoyl derivatives of selected (un) modified aminoalkanols A Gunia-Krzyżak, E Żesławska, K Słoczyńska, P Koczurkiewicz, W Nitek, ... European Journal of Medicinal Chemistry 107, 26-37, 2016 | 16 | 2016 |
| Chlorine substituents and linker topology as factors of 5-HT6R activity for novel highly active 1, 3, 5-triazine derivatives with procognitive properties in vivo S Sudoł, K Kucwaj-Brysz, R Kurczab, N Wilczyńska, ... European Journal of Medicinal Chemistry 203, 112529, 2020 | 15 | 2020 |
| The selenium-nitrogen bond as basis for reactive selenium species with pronounced antimicrobial activity J Rendekova, D Vlasakova, P Arsenyan, J Vasiljeva, MJ Nasim, K Witek, ... Current Organic Synthesis 14 (8), 1082-1090, 2017 | 15 | 2017 |
| Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy) alkyl]-and N-{2-[2-(phenoxy) ethoxy] ethyl} aminoalkanols as anticonvulsant agents AM Waszkielewicz, A Gunia-Krzyżak, B Powroźnik, K Słoczyńska, ... Bioorganic & Medicinal Chemistry 24 (8), 1793-1810, 2016 | 15 | 2016 |
| Seleno-vs. thioether triazine derivatives in search for new anticancer agents overcoming multidrug resistance in lymphoma W Ali, S Garbo, A Kincses, M Nové, G Spengler, E Di Bello, ... European Journal of Medicinal Chemistry 243, 114761, 2022 | 12 | 2022 |
| The synthesis and crystal structures of the homologues of epalrestat E Żesławska, W Nitek, W Tejchman Journal of Chemical Crystallography 45, 151-157, 2015 | 12 | 2015 |
| Phenylpiperazine 5,5-Dimethylhydantoin Derivatives as First Synthetic Inhibitors of Msr(A) Efflux Pump in Staphylococcus epidermidis K Witek, G Latacz, A Kaczor, J Czekajewska, E Żesławska, A Chudzik, ... Molecules 25 (17), 3788, 2020 | 11 | 2020 |
| Pharmacophoric features for a very potent 5‐spirofluorenehydantoin inhibitor of cancer efflux pump ABCB 1, based on X‐ray analysis E Żesławska, A Kincses, G Spengler, W Nitek, W Tejchman, J Handzlik Chemical Biology & Drug Design 93 (5), 844-853, 2019 | 11 | 2019 |
| Spectral Characteristic and Preliminary Anticancer Activity in vitro of Selected Rhodanine‐3‐carboxylic Acids Derivatives I Stawoska, W Tejchman, O Mazuryk, A Lyčka, P Nowak‐Sliwinska, ... Journal of Heterocyclic Chemistry 54 (5), 2889-2897, 2017 | 11 | 2017 |
| Amiloride conformation: The effect of different crystalline environments E Żesławska, B Oleksyn, K Stadnicka Structural Chemistry 15, 567-571, 2004 | 11 | 2004 |
